BioChemInsight: An Online Platform for Automated Extraction of Chemical Structures and Activity Data from Patents

Fuente: arXiv
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Autori principali: Wang, Zhe, Fu, Fangtian, Zhang, Wei, Yan, Lige, Li, Nan, Deng, Wenxia, Meng, Yan, Wu, Jianping, Wu, Hui, Wu, Wenting, Xu, Gang, Li, Xiang, Chen, Si
Natura: Preprint
Pubblicazione: 2025
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author Wang, Zhe
Fu, Fangtian
Zhang, Wei
Yan, Lige
Li, Nan
Deng, Wenxia
Meng, Yan
Wu, Jianping
Wu, Hui
Wu, Wenting
Xu, Gang
Li, Xiang
Chen, Si
author_facet Wang, Zhe
Fu, Fangtian
Zhang, Wei
Yan, Lige
Li, Nan
Deng, Wenxia
Meng, Yan
Wu, Jianping
Wu, Hui
Wu, Wenting
Xu, Gang
Li, Xiang
Chen, Si
contents The automated extraction of chemical structures and their corresponding bioactivity data is essential for accelerating drug discovery and enabling data-driven research. Current optical chemical structure recognition tools lack the capability to autonomously link molecular structures with their bioactivity profiles, posing a significant bottleneck in structure-activity relationship analysis. To address this, we present BioChemInsight, an open-source pipeline that integrates DECIMER Segmentation with MolNexTR for chemical structure recognition, GLM-4.5V for compound identifier association, and PaddleOCR combined with GLM-4.6 for bioactivity extraction and unit normalization. We evaluated BioChemInsight on 181 patents covering 15 therapeutic targets. The system achieved an average extraction accuracy of above 90% across three key tasks: chemical structure recognition, bioactivity data extraction, and compound identifier association. Our analysis indicates that the chemical space covered by patents is largely complementary to that contained in established public database ChEMBL. Consequently, by enabling systematic patent mining, BioChemInsight provides access to chemical information underrepresented in ChEMBL. This capability expands the landscape of explorable compound-target interactions, enriches the data foundation for quantitative structure-activity relationship modeling and targeted screening, and reduces data preprocessing time from weeks to hours. BioChemInsight is available at https://github.com/dahuilangda/BioChemInsight.
format Preprint
id arxiv_https___arxiv_org_abs_2504_10525
institution arXiv
publishDate 2025
record_format arxiv
spellingShingle BioChemInsight: An Online Platform for Automated Extraction of Chemical Structures and Activity Data from Patents
Wang, Zhe
Fu, Fangtian
Zhang, Wei
Yan, Lige
Li, Nan
Deng, Wenxia
Meng, Yan
Wu, Jianping
Wu, Hui
Wu, Wenting
Xu, Gang
Li, Xiang
Chen, Si
Quantitative Methods
Computation and Language
Information Retrieval
The automated extraction of chemical structures and their corresponding bioactivity data is essential for accelerating drug discovery and enabling data-driven research. Current optical chemical structure recognition tools lack the capability to autonomously link molecular structures with their bioactivity profiles, posing a significant bottleneck in structure-activity relationship analysis. To address this, we present BioChemInsight, an open-source pipeline that integrates DECIMER Segmentation with MolNexTR for chemical structure recognition, GLM-4.5V for compound identifier association, and PaddleOCR combined with GLM-4.6 for bioactivity extraction and unit normalization. We evaluated BioChemInsight on 181 patents covering 15 therapeutic targets. The system achieved an average extraction accuracy of above 90% across three key tasks: chemical structure recognition, bioactivity data extraction, and compound identifier association. Our analysis indicates that the chemical space covered by patents is largely complementary to that contained in established public database ChEMBL. Consequently, by enabling systematic patent mining, BioChemInsight provides access to chemical information underrepresented in ChEMBL. This capability expands the landscape of explorable compound-target interactions, enriches the data foundation for quantitative structure-activity relationship modeling and targeted screening, and reduces data preprocessing time from weeks to hours. BioChemInsight is available at https://github.com/dahuilangda/BioChemInsight.
title BioChemInsight: An Online Platform for Automated Extraction of Chemical Structures and Activity Data from Patents
topic Quantitative Methods
Computation and Language
Information Retrieval
url https://arxiv.org/abs/2504.10525