DMSO-promoted α-bromination of α-aryl ketones for the construction of 2-aryl-2-bromo-cycloketones.

Fuente: PubMed
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Autori principali: Zhai, Haojiang, Li, Penghui, Wang, Hongshuang, Wang, Xiaohui
Natura: Artículo científico
Lingua:en
Pubblicazione: Organic & biomolecular chemistry 2025
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author Zhai, Haojiang
Li, Penghui
Wang, Hongshuang
Wang, Xiaohui
author_facet Zhai, Haojiang
Li, Penghui
Wang, Hongshuang
Wang, Xiaohui
Zhai, Haojiang
Li, Penghui
Wang, Hongshuang
Wang, Xiaohui
collection PubMed - marine biology
contents DMSO-promoted α-bromination of α-aryl ketones for the construction of 2-aryl-2-bromo-cycloketones. Zhai, Haojiang Li, Penghui Wang, Hongshuang Wang, Xiaohui A DMSO-promoted practical one-step α-bromination reaction of α-aryl ketones with NBS has been developed for the construction of 2-aryl-2-bromo-cycloketones. The desired regioselective α-bromination products were isolated in moderate to good yields, with a maximum tested scale of 15 mmol. Notably, ketamine derivatives could be smoothly synthesized in two steps.
format Artículo científico
id pubmed_39760490
institution PubMed
language en
publishDate 2025
publisher Organic & biomolecular chemistry
record_format pubmed
spellingShingle DMSO-promoted α-bromination of α-aryl ketones for the construction of 2-aryl-2-bromo-cycloketones.
Zhai, Haojiang
Li, Penghui
Wang, Hongshuang
Wang, Xiaohui
DMSO-promoted α-bromination of α-aryl ketones for the construction of 2-aryl-2-bromo-cycloketones. Zhai, Haojiang Li, Penghui Wang, Hongshuang Wang, Xiaohui A DMSO-promoted practical one-step α-bromination reaction of α-aryl ketones with NBS has been developed for the construction of 2-aryl-2-bromo-cycloketones. The desired regioselective α-bromination products were isolated in moderate to good yields, with a maximum tested scale of 15 mmol. Notably, ketamine derivatives could be smoothly synthesized in two steps.
title DMSO-promoted α-bromination of α-aryl ketones for the construction of 2-aryl-2-bromo-cycloketones.
url https://pubmed.ncbi.nlm.nih.gov/39760490/