Actinomycetoquinones A-E, Anthraquinone-γ-Pyrones Discovered from Marine-Derived sp. Bacterium.

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Autori principali: Zhang, Fan, Roberts, Christopher D, Lee, Tae Hyun, Braun, Doug R, Bennett, Zachary D, Chanana, Shaurya, Guo, Song, Ananiev, Gene E, Guzei, Ilia A, Rajski, Scott R, Brunold, Thomas C, Bugni, Tim S
Natura: Artículo científico
Lingua:en
Pubblicazione: Journal of natural products 2025
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author Zhang, Fan
Roberts, Christopher D
Lee, Tae Hyun
Braun, Doug R
Bennett, Zachary D
Chanana, Shaurya
Guo, Song
Ananiev, Gene E
Guzei, Ilia A
Rajski, Scott R
Brunold, Thomas C
Bugni, Tim S
author_facet Zhang, Fan
Roberts, Christopher D
Lee, Tae Hyun
Braun, Doug R
Bennett, Zachary D
Chanana, Shaurya
Guo, Song
Ananiev, Gene E
Guzei, Ilia A
Rajski, Scott R
Brunold, Thomas C
Bugni, Tim S
Zhang, Fan
Roberts, Christopher D
Lee, Tae Hyun
Braun, Doug R
Bennett, Zachary D
Chanana, Shaurya
Guo, Song
Ananiev, Gene E
Guzei, Ilia A
Rajski, Scott R
Brunold, Thomas C
Bugni, Tim S
collection PubMed - marine biology
contents Actinomycetoquinones A-E, Anthraquinone-γ-Pyrones Discovered from Marine-Derived sp. Bacterium. Zhang, Fan Roberts, Christopher D Lee, Tae Hyun Braun, Doug R Bennett, Zachary D Chanana, Shaurya Guo, Song Ananiev, Gene E Guzei, Ilia A Rajski, Scott R Brunold, Thomas C Bugni, Tim S Anthraquinones Molecular Structure Pyrones Microbial Sensitivity Tests Anti-Bacterial Agents Methicillin-Resistant Staphylococcus aureus Escherichia coli Marine Biology Crystallography, X-Ray Actinobacteria Nuclear Magnetic Resonance, Biomolecular Facilitated by LC-MS-PCA metabolomics methods and effective molecular networking for strain prioritization and dereplication, five new anthraquinone-γ-pyrones, actinomycetoquinones A-E (-), were isolated from a marine-derived sp. bacterium. The structures of - were elucidated by analysis of their HRMS and NMR spectroscopic data. The absolute configuration of was unequivocally determined by single-crystal X-ray diffraction analysis using Cu Kα radiation. Actinomycetoquinone C exhibited antibacterial activity against methicillin-resistant (MRSA) and with MIC values of 1 and 4 μg/mL, respectively.
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language en
publishDate 2025
publisher Journal of natural products
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spellingShingle Actinomycetoquinones A-E, Anthraquinone-γ-Pyrones Discovered from Marine-Derived sp. Bacterium.
Zhang, Fan
Roberts, Christopher D
Lee, Tae Hyun
Braun, Doug R
Bennett, Zachary D
Chanana, Shaurya
Guo, Song
Ananiev, Gene E
Guzei, Ilia A
Rajski, Scott R
Brunold, Thomas C
Bugni, Tim S
Anthraquinones
Molecular Structure
Pyrones
Microbial Sensitivity Tests
Anti-Bacterial Agents
Methicillin-Resistant Staphylococcus aureus
Escherichia coli
Marine Biology
Crystallography, X-Ray
Actinobacteria
Nuclear Magnetic Resonance, Biomolecular
Actinomycetoquinones A-E, Anthraquinone-γ-Pyrones Discovered from Marine-Derived sp. Bacterium. Zhang, Fan Roberts, Christopher D Lee, Tae Hyun Braun, Doug R Bennett, Zachary D Chanana, Shaurya Guo, Song Ananiev, Gene E Guzei, Ilia A Rajski, Scott R Brunold, Thomas C Bugni, Tim S Anthraquinones Molecular Structure Pyrones Microbial Sensitivity Tests Anti-Bacterial Agents Methicillin-Resistant Staphylococcus aureus Escherichia coli Marine Biology Crystallography, X-Ray Actinobacteria Nuclear Magnetic Resonance, Biomolecular Facilitated by LC-MS-PCA metabolomics methods and effective molecular networking for strain prioritization and dereplication, five new anthraquinone-γ-pyrones, actinomycetoquinones A-E (-), were isolated from a marine-derived sp. bacterium. The structures of - were elucidated by analysis of their HRMS and NMR spectroscopic data. The absolute configuration of was unequivocally determined by single-crystal X-ray diffraction analysis using Cu Kα radiation. Actinomycetoquinone C exhibited antibacterial activity against methicillin-resistant (MRSA) and with MIC values of 1 and 4 μg/mL, respectively.
title Actinomycetoquinones A-E, Anthraquinone-γ-Pyrones Discovered from Marine-Derived sp. Bacterium.
topic Anthraquinones
Molecular Structure
Pyrones
Microbial Sensitivity Tests
Anti-Bacterial Agents
Methicillin-Resistant Staphylococcus aureus
Escherichia coli
Marine Biology
Crystallography, X-Ray
Actinobacteria
Nuclear Magnetic Resonance, Biomolecular
url https://pubmed.ncbi.nlm.nih.gov/40998300/