Development of Novel Protocol for Preclinical Monitoring the Release of Adjuvants Encapsulated Mucosal Delivery Carriers

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Autore principale: Mohamed Ibrahim-Saeed
Natura: Artículo científico
Lingua:en
Pubblicazione: Instituto Finlay 2015
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author Mohamed Ibrahim-Saeed
author_facet Mohamed Ibrahim-Saeed
contents Development of Novel Protocol for Preclinical Monitoring the Release of Adjuvants Encapsulated Mucosal Delivery Carriers Mohamed Ibrahim-Saeed Abd Rahaman-Omar Mohd Zobir-Hussein Isam Mohamed-Elkhidir Samer Hussein-Al-Ali Mothanna Sadiq-Al-Qubaisi Zamberi Sekawi Salud Nano adjuvant mucosal vaccines delivery carriers This work contributes in vaccines down-stream process by introducing a novel platform for in-vitro monitoring of vaccine-adjuvant delivery profile as a crucial preclinical optimizing step in mucosal vaccines. Nano and micro particles of Calcium phosphate (Cap) vaccine-adjuvant were encapsulated in Chitosan and Alginate polymeric carriers. Adjuvants release profiles monitored in a permeable bag at 37°C, pH 2, incubated in isotonic buffer for 96 hours. The released Calcium in the outer buffer was monitored and compared in-addition to the carrier’s swelling and biophysical properties. The adjuvants and carriers did not interfere with the proliferation of cultured hepatocytes an indicator of their safe use; Chitosan’s viscosity and swelling were higher than Alginate. Chitosan’s Zeta-potential was significantly high positive, while Cap and Alginate were negative. The prepared CaP and Chitosan particles were in nano-size, while the ready-made CaP adjuvant and Alginate were in micro-size using zeta-seizer and scanning electron-micrograph. The release of nano-size particle was in ascending, extended and controlled manner compared to micro-size adjuvant. Moreover, nano-adjuvant release profile from Chitosan was superior compared to Alginate. The core controlling factors in vaccine-adjuvant sustained release includes; smaller adjuvant particles (nano-size), carrier’s low swelling, high viscosity and importantly carrier-adjuvant entrapment reversibility. Chitosan offers sustained ascending superior capacity in releasing Nano-Cap adjuvant. This novel in-vitro pre-clinical study answer a crucial downstream preparative step for optimizing mucosal vaccines before their direct routine in-vivo trial on animal regardless of adjuvant’s particle size or delivery kinetics. 2015 artículo científico 1025-0298 https://www.redalyc.org/articulo.oa?id=203443342004 en http://www.redalyc.org/revista.oa?id=2034 VacciMonitor application/pdf Instituto Finlay VacciMonitor (Cuba) Num.3 Vol.24
format Artículo científico
id redalyc_203443342004
language en
publishDate 2015
publisher Instituto Finlay
spellingShingle Development of Novel Protocol for Preclinical Monitoring the Release of Adjuvants Encapsulated Mucosal Delivery Carriers
Mohamed Ibrahim-Saeed
Salud
Nano
adjuvant
mucosal vaccines
delivery carriers
Development of Novel Protocol for Preclinical Monitoring the Release of Adjuvants Encapsulated Mucosal Delivery Carriers Mohamed Ibrahim-Saeed Abd Rahaman-Omar Mohd Zobir-Hussein Isam Mohamed-Elkhidir Samer Hussein-Al-Ali Mothanna Sadiq-Al-Qubaisi Zamberi Sekawi Salud Nano adjuvant mucosal vaccines delivery carriers This work contributes in vaccines down-stream process by introducing a novel platform for in-vitro monitoring of vaccine-adjuvant delivery profile as a crucial preclinical optimizing step in mucosal vaccines. Nano and micro particles of Calcium phosphate (Cap) vaccine-adjuvant were encapsulated in Chitosan and Alginate polymeric carriers. Adjuvants release profiles monitored in a permeable bag at 37°C, pH 2, incubated in isotonic buffer for 96 hours. The released Calcium in the outer buffer was monitored and compared in-addition to the carrier’s swelling and biophysical properties. The adjuvants and carriers did not interfere with the proliferation of cultured hepatocytes an indicator of their safe use; Chitosan’s viscosity and swelling were higher than Alginate. Chitosan’s Zeta-potential was significantly high positive, while Cap and Alginate were negative. The prepared CaP and Chitosan particles were in nano-size, while the ready-made CaP adjuvant and Alginate were in micro-size using zeta-seizer and scanning electron-micrograph. The release of nano-size particle was in ascending, extended and controlled manner compared to micro-size adjuvant. Moreover, nano-adjuvant release profile from Chitosan was superior compared to Alginate. The core controlling factors in vaccine-adjuvant sustained release includes; smaller adjuvant particles (nano-size), carrier’s low swelling, high viscosity and importantly carrier-adjuvant entrapment reversibility. Chitosan offers sustained ascending superior capacity in releasing Nano-Cap adjuvant. This novel in-vitro pre-clinical study answer a crucial downstream preparative step for optimizing mucosal vaccines before their direct routine in-vivo trial on animal regardless of adjuvant’s particle size or delivery kinetics. 2015 artículo científico 1025-0298 https://www.redalyc.org/articulo.oa?id=203443342004 en http://www.redalyc.org/revista.oa?id=2034 VacciMonitor application/pdf Instituto Finlay VacciMonitor (Cuba) Num.3 Vol.24
title Development of Novel Protocol for Preclinical Monitoring the Release of Adjuvants Encapsulated Mucosal Delivery Carriers
topic Salud
Nano
adjuvant
mucosal vaccines
delivery carriers
url https://www.redalyc.org/articulo.oa?id=203443342004