Copertina

Design and Synthesis of Potent Ridaifen Analogues: Evaluation as Anticancer, 20S Proteasomal Inhibitors, and Antiebola Virus Agents through In vitro and In Silico Studies

Fuente: Wiley Open Access

Salvato in:

Dettagli Bibliografici
Autori principali:	Merna A. Vector, Sae Fujiwara, Yunhao Zhu, Makoto Hasegawa, Takatsugu Murata, Kaho Tsuchiya, Isamu Shiina, Ashraf H. Abadi, Nermin S. Ahmed
Natura:	Artículo Open Access
Pubblicazione:	Wiley 2025
Soggetti:	ChemMedChem
Accesso online:	Acceder al recurso
Tags:	Aggiungi Tag Nessun Tag, puoi essere il primo ad aggiungerne!!

Documenti analoghi

Sphaeropsidin A C15–C16 Cross‐Metathesis Analogues with Potent Anticancer Activity
di: Sachin B. Wagh, et al.
Pubblicazione: (2024)

In Silico‐Enabled Discovery and Development of Potent and Selective CDK11 Inhibitors
di: Frankie S. Mak, et al.
Pubblicazione: (2026)

Design, Synthesis, and In Vitro and In Silico Anticancer Profiling of Spirooxindole–Tetrahydrocarbazoles
di: Supriya Sharma, et al.
Pubblicazione: (2026)

Exploration of the Anticancer Efficacy and In Silico Drug Screening Study of Fe(II) and Fe(III) Complexes of Schiff Base and Phenanthroline Ligand
di: Jansi Rani J, et al.
Pubblicazione: (2026)

Front Cover: Functional Proteomics of Quinazolin‐4‐One Derivatives Targeting the Proteasome (ChemMedChem 2/2026)
di: Elva Morretta, et al.
Pubblicazione: (2026)

Artificial Ion Transporters as Potent Therapeutics for Channelopathies
di: Wei Huang, et al.
Pubblicazione: (2024)

GDF15 Analogues Acting as GFRAL Ligands
di: Andrea Di Santo, et al.
Pubblicazione: (2025)

2‐Carboxyquinoline Boronic Acids as Highly Potent KPC Inhibitors
di: Zheng Ma, et al.
Pubblicazione: (2025)

Development of Novel Anticancer Pyrazolopyrimidinones Targeting Glioblastoma
di: Kate Byrne, et al.
Pubblicazione: (2025)

Sulphur Analogues of Homoisoflavonoids as Potential Treatments for Neovascular Eye Diseases
di: Jacob D. Hiles, et al.
Pubblicazione: (2026)

Diversity Oriented Synthesis of Novel Xanthones Reveal Potent Doxorubicin‐Inspired Analogs
di: Jonas W. Meringdal, et al.
Pubblicazione: (2024)

Synthesis and Evaluation of Fluorinated Piperazine‐Hydroxyethylamine Analogues as Potential Antiplasmodial Candidates
di: Charu Upadhyay, et al.
Pubblicazione: (2024)

Isoflavone Derivatives as Potential Anticancer Agents: Synthesis and Bioactivity Studies
di: Mamoalosi A. Selepe
Pubblicazione: (2024)

Modified Nucleotides in Bifunctional Antisense Oligonucleotides: Exploring their Anticancer Potential
di: Natalia Bartyś, et al.
Pubblicazione: (2025)

Exploring Small‐Molecule Modulators of Precursor miRNA Processing Associated With Glycolysis
di: Miho Fujiki, et al.
Pubblicazione: (2026)

Bushy‐Tailed Multicationic Quaternary Phosphonium Compounds: Potent Amphiphilic Disinfectants with Promising Therapeutic Indices
di: Diana Rachii, et al.
Pubblicazione: (2024)

Tryptophan‐Rich Short Peptide Amphiphile‐Mediated Synthesis of Silver Nanoparticles for Potent Antibacterial Applications
di: Govind Singh, et al.
Pubblicazione: (2025)

4‐Aza Cyclopentenone Prostaglandin Analogues: Synthesis and NF‐κB Inhibitory Activities
di: William Doherty, et al.
Pubblicazione: (2024)

Small Molecule‐Drug Conjugates: Opportunities for the Development of Targeted Anticancer Drugs
di: Jingjing Zhang, et al.
Pubblicazione: (2024)

Efficacy of DNA Intercalator‐Conjugated Triplex‐Forming Oligonucleotide as Anticancer Agent
di: Haruki Toyama, et al.
Pubblicazione: (2025)

Lactam Truncation Yields a Dihydroquinazolinone Scaffold with Potent Antimalarial Activity that Targets PfATP4
di: Trent D. Ashton, et al.
Pubblicazione: (2024)

Potent Antisickling Furaldehyde Analogs for Acute Sickle Cell Therapy: Enhanced Efficacy and Intravenous Formulation Potential
di: Abdelsattar M. Omar, et al.
Pubblicazione: (2025)

Discovery of Potent Isoindolinone Inhibitors that Target an Active Conformation of PARP1 Using DNA‐Encoded Libraries
di: Kelly A. McCarthy, et al.
Pubblicazione: (2024)

Design and Synthesis of Novel β‐Carboline‐Bisindole Hybrids as Potential Anticancer Agents
di: Nguyen Thi Thanh Huyen, et al.
Pubblicazione: (2024)

Strategic Design and Development of Indole‐Based Compounds as Potent Malic Enzyme 3 Inhibitors for Pancreatic Tumor Therapy
di: Gaurav Sheth, et al.
Pubblicazione: (2025)

An Internal Sulfur–Lone Pair Interaction Enabled the Discovery of Potent and Sub‐Family Selective PKMYT1 Inhibitors
di: Yazhou Wang, et al.
Pubblicazione: (2026)

Preparation of Dearomatized p‐Coumaric Acid Derivatives as DNA Damage Response Inhibitors with Potent In Vitro Antitumor Effect
di: Laura Fási, et al.
Pubblicazione: (2024)

In Silico Prediction of ERRα Agonists Based on Combined Features and Stacking Ensemble Method
di: Jiahao Xu, et al.
Pubblicazione: (2024)

Design and Synthesis of 2‐Nitroimidazole‐1,2,3‐triazole Sulfonamide Hybrids as Potent and Selective Anti‐Trypanosomatid Agents
di: Victória C. Tietz, et al.
Pubblicazione: (2024)

Development of Carborane‐Based Halogenated Naphthyridinone‐Analogues as Cannabinoid Receptor Type 2 (CB 2 R) Ligands
di: Lea Ueberham, et al.
Pubblicazione: (2025)

Design and Synthesis of Pyrimidino[4,5‐ d ]Pyrimidine‐Based Compounds as Potent B‐RAF V600E Inhibitors
di: Eleftheria A. Georgiou, et al.
Pubblicazione: (2026)

Discovery of Galactopyranose‐1‐carboxamides as a New Class of Small, Novel, Potent, Selective, and Orally Active Galectin‐3 Inhibitors
di: Cornelia Zumbrunn, et al.
Pubblicazione: (2025)

Advances in Diclofenac Derivatives: Exploring Carborane‐Substituted N‐Methyl and Nitrile Analogs for Anticancer Therapy
di: Christoph Selg, et al.
Pubblicazione: (2025)

In Vitro and In Vivo Biological Evaluation of Novel 1,4‐Naphthoquinone Derivatives as Potential Anticancer Agents
di: Palanisamy Ravichandiran, et al.
Pubblicazione: (2024)

Next‐Generation Bcl‐2 Inhibitors: Design and Evaluation of Indolyl‐Triazole Derivatives with Anticancer Potential
di: Ahmed M. Almehdi, et al.
Pubblicazione: (2025)

CORRIGENDUM: Carboranes as Potent Phenyl Mimetics: A Comparative Study on the Reversal of ABCG2‐Mediated Drug Resistance by Carboranylquinazolines and Their Organic Isosteres
Pubblicazione: (2024)

Design and Synthesis of Sulfonium and Selenonium Derivatives Bearing 3′,5′‐ O ‐Benzylidene Acetal Side Chains as Potent α ‐Glucosidase Inhibitors
di: Yaojia Li, et al.
Pubblicazione: (2025)

Cytotoxic, Antibacterial, and in Silico Pks13 Inhibitory Properties of Indole‐Coupled Dihydrobenzo[c]phenanthridines
di: Reyna Martha Gallegos‐Alvarado, et al.
Pubblicazione: (2025)

Chemical Derivatization Leads to the Discovery Of Novel Analogs of Azotochelin, a Natural Siderophore, as Promising Anticancer Agents
di: Nishant M. Karadkhelkar, et al.
Pubblicazione: (2024)

Synthesis And Anticancer Activity Of New Hybrid 3‐Methylidene‐2,3‐Dihydro‐1,8‐Naphthyridinones
di: Agata Jaskulska, et al.
Pubblicazione: (2024)